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Exploring Potential of 1,5-Benzothiazepines: A Brief Review


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1 Department of Pharmaceutical Chemistry, Y.B. Chavan College of Pharmacy. Dr. Rafiq Zakaria Campus, Aurangabad. 431001.(MS), India
     

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Benzothiazepines are fused heterocyclic compounds. They are claimed of various therapeutic activities and hence, they are utilized in drug research. Recently, attention is being directed to their synthetic methods, chemical and biological properties. Benzothiazepines posses wide variety of biological activities like anticonvulsant, CNS depressant, Ca++ channel blockers, calcium channel modulator, calcium channel antagonist, anticancer, anti fungal antimicrobial, anti‐HIV and anti-anginal.

Keywords

1,5-benzothiazepine, CNS, Green Synthesis, Microwave –assisted
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Abstract Views: 279

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  • Exploring Potential of 1,5-Benzothiazepines: A Brief Review

Abstract Views: 279  |  PDF Views: 3

Authors

A. P. G Nikalje
Department of Pharmaceutical Chemistry, Y.B. Chavan College of Pharmacy. Dr. Rafiq Zakaria Campus, Aurangabad. 431001.(MS), India
M. Ghodke
Department of Pharmaceutical Chemistry, Y.B. Chavan College of Pharmacy. Dr. Rafiq Zakaria Campus, Aurangabad. 431001.(MS), India
S. Tiwari
Department of Pharmaceutical Chemistry, Y.B. Chavan College of Pharmacy. Dr. Rafiq Zakaria Campus, Aurangabad. 431001.(MS), India

Abstract


Benzothiazepines are fused heterocyclic compounds. They are claimed of various therapeutic activities and hence, they are utilized in drug research. Recently, attention is being directed to their synthetic methods, chemical and biological properties. Benzothiazepines posses wide variety of biological activities like anticonvulsant, CNS depressant, Ca++ channel blockers, calcium channel modulator, calcium channel antagonist, anticancer, anti fungal antimicrobial, anti‐HIV and anti-anginal.

Keywords


1,5-benzothiazepine, CNS, Green Synthesis, Microwave –assisted

References